pregabalina
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Pregabalina is a GABA analogous, although it does not bind to its receptor and is not able to develop characteristic actions. | PGBB es un análogo del GABA aunque no se liga a su receptor, ni es capaz de desarrollar acciones gabaérgicas. |
Pregabalina does not bind to plasma proteins and it has intact elimination almost totality, that is why it presents tiny interaction with other drugs. | PGBB no se liga a las proteínas plasmáticas y se elimina inalterada por orina casi en su totalidad, por lo que presenta escasa interacción con otros fármacos. |
In all pain animals' models, 150 mg of Pregabalina at day or superior has demonstrated to be more effectiveness than placebo, just with a dose-dependent form to control pain, to improve sleep and life's quality of patients. | En todos ellos, PGBB en dosis de 150 mg. día o superiores, ha demostrado eficacia frente a placebo de una forma dosis dependiente para controlar el dolor, mejorar el sueño y mejorar muchos de los parámetros de la calidad de vida de los pacientes. |
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